Novel SARS-CoV-2 inhibition properties of the anti-cancer Kang Guan Recipe herbal formula

Cancer Lett. 2024 Nov 1:604:217198. doi: 10.1016/j.canlet.2024.217198. Epub 2024 Aug 27.

Abstract

The ongoing COVID-19 pandemic is a persistent challenge, with continued breakthrough infections despite vaccination efforts. This has spurred interest in alternative preventive measures, including dietary and herbal interventions. Previous research has demonstrated that herbal medicines can not only inhibit cancer progression but also combat viral infections, including COVID-19 by targeting SARS-CoV-2, indicating a multifaceted potential to address both viruses and cancer. Here, we found that the Kang Guan Recipe (KGR), a novel herbal medicine formula, associates with potent inhibition activity against the SARS-CoV-2 viral infection. We demonstrate that KGR exhibits inhibitory activity against several SARS-CoV-2 variants of concern (VOCs). Mechanistically, we found that KGR can block the interaction of the viral spike and human angiotensin-converting enzyme 2 (ACE2). Furthermore, we assessed the inhibitory effect of KGR on SARS-CoV-2 viral entry in vivo, observing that serum samples from healthy human subjects having taken KGR exhibited suppressive activity against SARS-CoV-2 variants. Our investigation provides valuable insights into the potential of KGR as a novel herbal-based preventive and therapeutic strategy against COVID-19.

Keywords: Angiotensin-converting enzyme 2; Coronavirus disease 2019; Kang guan recipe; Severe acute respiratory syndrome coronavirus 2; Variants of concern.

MeSH terms

  • Angiotensin-Converting Enzyme 2* / antagonists & inhibitors
  • Angiotensin-Converting Enzyme 2* / metabolism
  • Animals
  • Antiviral Agents / pharmacology
  • COVID-19 / prevention & control
  • COVID-19 / virology
  • COVID-19 Drug Treatment
  • Chlorocebus aethiops
  • Drugs, Chinese Herbal* / pharmacology
  • Humans
  • SARS-CoV-2* / drug effects
  • Spike Glycoprotein, Coronavirus* / metabolism
  • Vero Cells
  • Virus Internalization* / drug effects

Substances

  • Angiotensin-Converting Enzyme 2
  • Drugs, Chinese Herbal
  • Spike Glycoprotein, Coronavirus
  • Antiviral Agents
  • ACE2 protein, human
  • spike protein, SARS-CoV-2

Supplementary concepts

  • SARS-CoV-2 variants