Exposure to endocrine disruptor DEHP promotes the progression and radiotherapy resistance of pancreatic cancer cells by increasing BMI1 expression and properties of cancer stem cells

Ecotoxicol Environ Saf. 2024 Sep 15:283:116970. doi: 10.1016/j.ecoenv.2024.116970. Epub 2024 Aug 30.

Abstract

Most patients diagnosed with pancreatic cancer are initially at an advanced stage, and radiotherapy resistance impact the effectiveness of treatment. This study aims to investigate the effects of endocrine disruptor Di-(2-ethylhexyl) phthalate (DEHP) on various biological behaviors and the radiotherapy sensitivity of pancreatic cancer cells, as well as its potential mechanisms. Our findings indicate that exposure to DEHP promotes the proliferation of various cancer cells, including those from the lung, breast, pancreas, and liver, in a time- and concentration-dependent manner. Furthermore, DEHP exposure could influence several biological behaviors of pancreatic cancer cells in vivo and vitro. These effects include reducing cell apoptosis, causing G0/G1 phase arrest, increasing migration capacity, enhancing tumorigenicity, elevating the proportion of cancer stem cells (CSCs), and upregulating expression levels of CSCs markers such as CD133 and BMI1. DEHP exposure can also increase radiation resistance, which can be reversed by downregulating BMI1 expression. In summary our research suggests that DEHP exposure can lead to pancreatic cancer progression and radiotherapy resistance, and the mechanism may be related to the upregulation of BMI1 expression, which leads to the increase of CSCs properties.

Keywords: Cancer stem cells; DEHP; Endocrine disruptor; Pancreatic cancer; Radiotherapy resistance.

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Apoptosis / radiation effects
  • Cell Line, Tumor
  • Cell Movement / drug effects
  • Cell Movement / radiation effects
  • Cell Proliferation / drug effects
  • Cell Proliferation / radiation effects
  • Diethylhexyl Phthalate* / toxicity
  • Disease Progression
  • Endocrine Disruptors* / toxicity
  • Humans
  • Mice
  • Mice, Nude
  • Neoplastic Stem Cells* / drug effects
  • Neoplastic Stem Cells* / radiation effects
  • Pancreatic Neoplasms* / pathology
  • Polycomb Repressive Complex 1 / genetics
  • Polycomb Repressive Complex 1 / metabolism
  • Radiation Tolerance* / drug effects

Substances

  • Diethylhexyl Phthalate
  • Endocrine Disruptors
  • Polycomb Repressive Complex 1
  • BMI1 protein, human