The role of high mobility group box-1 on the development of diabetes complications: A plausible pharmacological target

Diab Vasc Dis Res. 2024 Sep-Oct;21(5):14791641241271949. doi: 10.1177/14791641241271949.

Abstract

Background: Diabetes mellitus has emerged as a pressing global concern, with a notable increase in recent years. Despite advancements in treatment, existing medications struggle to halt the progression of diabetes and its associated complications. Increasing evidence underscores inflammation as a significant driver in the onset of diabetes mellitus. Therefore, perspectives on new therapies must consider shifting focus from metabolic stress to inflammation. High mobility group box (HMGB-1), a nuclear protein regulating gene expression, gained attention as an endogenous danger signal capable of sparking inflammatory responses upon release into the extracellular environment in the late 1990s.

Purpose: Given the parallels between inflammatory responses and type 2 diabetes (T2D) development, this review paper explores HMGB-1's potential involvement in onset and progression of diabetes complications. Specifically, we will review and update the understanding of HMGB-1 and its inflammatory pathways in insulin resistance, diabetic nephropathy, diabetic neuropathy, and diabetic retinopathy.

Conclusions: HMGB-1 and its receptors i.e. receptor for advanced glycation end-products (RAGE) and toll-like receptors (TLRs) present promising targets for antidiabetic interventions. Ongoing and future projects in this realm hold promise for innovative approaches targeting HMGB-1-mediated inflammation to ameliorate diabetes and its complications.

Keywords: HMGB-1; diabetes complications; diabetic nephropathy; diabetic neuropathy; diabetic retinopathy.

Publication types

  • Review

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / therapeutic use
  • Diabetes Complications / drug therapy
  • Diabetes Complications / metabolism
  • Diabetes Mellitus, Type 2 / drug therapy
  • Diabetes Mellitus, Type 2 / metabolism
  • Diabetic Nephropathies / drug therapy
  • Diabetic Nephropathies / metabolism
  • Diabetic Neuropathies / drug therapy
  • Diabetic Neuropathies / etiology
  • Diabetic Neuropathies / metabolism
  • Diabetic Retinopathy / drug therapy
  • Diabetic Retinopathy / etiology
  • Diabetic Retinopathy / metabolism
  • Diabetic Retinopathy / prevention & control
  • HMGB1 Protein* / antagonists & inhibitors
  • HMGB1 Protein* / metabolism
  • Humans
  • Hypoglycemic Agents* / therapeutic use
  • Inflammation Mediators / metabolism
  • Insulin Resistance
  • Molecular Targeted Therapy
  • Receptor for Advanced Glycation End Products* / antagonists & inhibitors
  • Receptor for Advanced Glycation End Products* / metabolism
  • Signal Transduction*
  • Toll-Like Receptors / metabolism

Substances

  • HMGB1 Protein
  • Receptor for Advanced Glycation End Products
  • HMGB1 protein, human
  • Hypoglycemic Agents
  • Inflammation Mediators
  • Anti-Inflammatory Agents
  • Toll-Like Receptors