Endomorphin-2 (Endo2) and substance P (SubP) co-application attenuates SubP-induced excitation and alters frequency plasticity in neonatal rat in vitro preparations

Respir Physiol Neurobiol. 2025 Jan:331:104351. doi: 10.1016/j.resp.2024.104351. Epub 2024 Sep 19.

Abstract

Substance P (SubP) and endomorphin-2 (Endo2) are co-localized presynaptically in vesicles of neurons adjacent to inspiratory rhythm-generating pre-Botzinger Complex (preBotC) neurons but the effects of co-released SubP and Endo2 on respiratory motor control are not known. To address this question, SubP alone or a combination of SubP and Endo2 (SubP/Endo2) were bath-applied in a sustained (15-min) or intermittent (5-min application, 5-min washout, x3) pattern at 10-100 nM to neonatal rat brainstem-spinal cord preparations. During neuropeptide application, SubP/Endo2 co-applications generally attenuated SubP-induced increases in burst frequency and decreases in burst amplitude. With respect to frequency plasticity (long-lasting increase in burst frequency 60 min post-neuropeptide application), SubP-induced frequency plasticity was increased with sustained SubP/Endo2 co-applications at 20 and 100 nM. Intermittent SubP/Endo2 co-applications tended to decrease the level of frequency plasticity induced by intermittent SubP alone applications. SubP/Endo2 co-applications revealed potentially new functions for neurokinin-1 (NK1R) and mu-opioid (MOR) receptors on respiratory rhythm-generating medullary neurons.

Keywords: Mu-opioid receptor; Neonatal rat; Neurokinin-1 receptor; Neuromodulation; Neuroplasticity; Respiratory motor control.

MeSH terms

  • Action Potentials / drug effects
  • Action Potentials / physiology
  • Animals
  • Animals, Newborn*
  • Brain Stem* / drug effects
  • Brain Stem* / physiology
  • Dose-Response Relationship, Drug
  • In Vitro Techniques
  • Neuronal Plasticity* / drug effects
  • Neuronal Plasticity* / physiology
  • Neurons / drug effects
  • Neurons / physiology
  • Oligopeptides* / administration & dosage
  • Oligopeptides* / pharmacology
  • Rats
  • Rats, Sprague-Dawley*
  • Spinal Cord* / drug effects
  • Spinal Cord* / physiology
  • Substance P* / pharmacology

Substances

  • Substance P
  • Oligopeptides
  • endomorphin 2