Nanoparticle-Directed Antioxidant Therapy Can Ameliorate Disease Progression in a Novel, Diet-Inducible Model of Coronary Artery Disease

Arterioscler Thromb Vasc Biol. 2024 Dec;44(12):2476-2488. doi: 10.1161/ATVBAHA.124.321030. Epub 2024 Oct 17.

Abstract

Background: Oxidative stress plays a crucial role in the pathogenesis of coronary artery disease. In cardiovascular research using murine models, the generation and maintenance of models with robust coronary arterial atherosclerosis has been challenging.

Methods: We characterized a new mouse model in which the last 3 amino acids of the carboxyl terminus of the HDL (high-density lipoprotein) receptor (SR-B1 [scavenger receptor, class B, type 1]) were deleted in a low-density lipoprotein receptor knockout (LDLR-/-) mouse model (SR-B1ΔCT/LDLR-/-) fed an atherogenic diet. We also tested the therapeutic effects of an oxidative stress-targeted nanoparticle in atherogenic diet-fed SR-B1ΔCT/LDLR-/- mice.

Results: The SR-B1ΔCT/LDLR-/- mice fed an atherogenic diet had occlusive coronary artery atherosclerosis, impaired cardiac function, and a dramatically lower survival rate, compared with LDLR-/- mice fed the same diet. As SR-B1ΔCT/LDLR-/- mice do not exhibit female infertility or low pup yield, they are far easier and less costly to use than the previously described SR-B1-based models of coronary artery disease. We found that treatment with the targeted nanoparticles improved the cardiac functions and corrected hematologic abnormalities caused by the atherogenic diet in SR-B1ΔCT/LDLR-/- mice but did not alter the distinctive plasma lipid levels.

Conclusions: The SR-B1ΔCT/LDLR-/- mice developed diet-inducible, fatal atherosclerotic coronary artery disease, which could be ameliorated by targeted nanoparticle therapy. Our study provides new tools for the development of cardiovascular therapies.

Keywords: diet, atherogenic; high-density lipoprotein receptors; mice, knockout; survival rate.

MeSH terms

  • Animals
  • Antioxidants* / administration & dosage
  • Antioxidants* / pharmacology
  • Coronary Artery Disease* / drug therapy
  • Coronary Artery Disease* / genetics
  • Coronary Artery Disease* / metabolism
  • Coronary Artery Disease* / pathology
  • Coronary Artery Disease* / prevention & control
  • Diet, Atherogenic / adverse effects
  • Disease Models, Animal*
  • Disease Progression*
  • Female
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout*
  • Nanoparticles*
  • Oxidative Stress* / drug effects
  • Receptors, LDL* / deficiency
  • Receptors, LDL* / genetics
  • Scavenger Receptors, Class B* / deficiency
  • Scavenger Receptors, Class B* / genetics
  • Scavenger Receptors, Class B* / metabolism

Substances

  • Receptors, LDL
  • Antioxidants
  • Scavenger Receptors, Class B
  • Scarb1 protein, mouse