Improved Localization of Insulinomas Using 68Ga-NODAGA-Exendin-4 PET/CT

J Nucl Med. 2024 Dec 3;65(12):1959-1964. doi: 10.2967/jnumed.124.268158.

Abstract

Precise anatomic localization of insulinomas is crucial for surgical treatment. Current routine noninvasive imaging techniques, including CT, MRI, and 68Ga-DOTA-somatostatin analog (DOTA-SSA) PET/CT, have limited sensitivity. Endoscopic ultrasound is highly sensitive but invasive. In this prospective multicenter study, we compared the diagnostic accuracy of 68Ga-NODAGA-exendin-4 (exendin) PET/CT with all routine imaging procedures for the localization of insulinomas. Methods: Sixty-nine adults with biochemically proven adult endogenous hyperinsulinemic hypoglycemia underwent exendin PET/CT and current routine imaging. Images were evaluated in a clinical reading and in an expert reading. Image quality was determined by quantitative analysis. Results: Based on clinical readings, the accuracy of exendin PET/CT (94.4%; 95% CI, 84.6%-98.8%) was greater than that of DOTA-SSA PET/CT (64.8%; 95% CI, 50.6%-77.3%), contrast-enhanced CT/contrast-enhanced diffusion-weighted imaging-MRI (83.3%; 95% CI, 70.7%-92.1%), and endoscopic ultrasound (82.8%; 95% CI, 64.1%-94.1%). In 13% of patients, a correct diagnosis was only reached after exendin PET/CT. Interobserver agreement between readings was higher for exendin PET/CT than for DOTA-SSA PET/CT and contrast-enhanced CT/contrast-enhanced diffusion-weighted imaging-MRI (Cohen κ, 1.0 vs. 0.5 and 0.55). Exendin PET/CT provided a higher insulinoma-to-background ratio (15.3 ± 6.7 vs. 5.2 ± 3.0) and contrast-to-noise ratio (22.6 ± 11.1 vs. 5.1 ± 3.7) than did DOTA-SSA PET/CT. Conclusion: This study demonstrates the superiority of exendin PET/CT in a unique prospective comparison to all current routine imaging modalities for preoperative localization of benign insulinomas, providing the level of evidence needed for clinical implementation.

Keywords: GLP-1 receptor; diagnostic imaging; exendin PET/CT; insulinoma.

Publication types

  • Multicenter Study

MeSH terms

  • Acetates / chemistry
  • Adult
  • Aged
  • Exenatide*
  • Female
  • Gallium Radioisotopes*
  • Heterocyclic Compounds, 1-Ring* / chemistry
  • Humans
  • Insulinoma* / diagnostic imaging
  • Male
  • Middle Aged
  • Pancreatic Neoplasms / diagnostic imaging
  • Peptides / chemistry
  • Positron Emission Tomography Computed Tomography*
  • Prospective Studies
  • Radiopharmaceuticals
  • Venoms / chemistry

Substances

  • Exenatide
  • Heterocyclic Compounds, 1-Ring
  • 1-(1,3-carboxypropyl)-4,7-carboxymethyl-1,4,7-triazacyclononane
  • Gallium Radioisotopes
  • Acetates
  • Peptides
  • Venoms
  • Radiopharmaceuticals