Metabolic Syndrome Nonalcoholic Steatohepatitis Male Mouse With Adeno-Associated Viral Renin as a Novel Model for Heart Failure With Preserved Ejection Fraction

J Am Heart Assoc. 2024 Dec 3;13(23):e035894. doi: 10.1161/JAHA.124.035894. Epub 2024 Nov 22.

Abstract

Background: Heart failure with preserved ejection fraction (HFpEF) currently accounts for more than half of patients with HF, with limited approved evidence-based therapies. HFpEF is a complex multifactorial disease associated with hypertension, obesity, diabetes, and renal dysfunction. In addition to our limited understanding of HFpEF pathophysiology, the development of new therapies is partially hindered by the existing translationally relevant preclinical HFpEF models.

Methods and results: Here, we report the development of a novel 2-hit HFpEF male mouse model through adding hypertensive stress from the activation of the renin-angiotensin-aldosterone system with adeno-associated viral-renin (AAV-renin), to the metabolic syndrome nonalcoholic steatohepatitis (MSNASH, formerly FATZO) mouse (MSNASH+AAV-renin). To further demonstrate model translatability, MSNASH+AAV-renin mice were then treated with approved HFpEF therapies sacubitril/valsartan or a combination of sacubitril/valsartan and empagliflozin. We found that the MSNASH+AAV-renin mouse model demonstrates clinically relevant features of human HFpEF, including preserved ejection fraction, cardiac hypertrophy, left atrial enlargement, diastolic dysfunction, elevated natriuretic peptides, inflammation, and low exercise capacity. We also demonstrate that treatment with approved HFpEF therapies sacubitril/valsartan and the combination of sacubitril/valsartan with empagliflozin improves the cardiac phenotypes of HFpEF in this model.

Conclusions: The MSNASH+AAV-renin model faithfully represents a severe cardiometabolic HFpEF phenogroup that can be used as a new tool for HFpEF preclinical research and drug discovery.

Keywords: HFpEF; MSNASH; cardiometabolism; empagliflozin; mouse models; renin; sacubitril/valsartan.

MeSH terms

  • Aminobutyrates / pharmacology
  • Angiotensin Receptor Antagonists / pharmacology
  • Angiotensin Receptor Antagonists / therapeutic use
  • Animals
  • Benzhydryl Compounds / pharmacology
  • Benzhydryl Compounds / therapeutic use
  • Biphenyl Compounds
  • Dependovirus* / genetics
  • Disease Models, Animal*
  • Drug Combinations
  • Genetic Vectors
  • Heart Failure* / metabolism
  • Heart Failure* / physiopathology
  • Male
  • Metabolic Syndrome* / complications
  • Metabolic Syndrome* / physiopathology
  • Mice
  • Mice, Inbred C57BL
  • Non-alcoholic Fatty Liver Disease* / metabolism
  • Non-alcoholic Fatty Liver Disease* / physiopathology
  • Renin* / blood
  • Renin* / metabolism
  • Renin-Angiotensin System* / physiology
  • Stroke Volume*
  • Tetrazoles / pharmacology
  • Valsartan*
  • Ventricular Function, Left

Substances

  • Renin
  • Valsartan
  • Aminobutyrates
  • sacubitril and valsartan sodium hydrate drug combination
  • Drug Combinations
  • Biphenyl Compounds
  • Tetrazoles
  • Benzhydryl Compounds
  • Angiotensin Receptor Antagonists