Synthesis of Pentafluorosulfanylated Ynamides and Further Functionalizations

Org Lett. 2024 Dec 6;26(48):10369-10375. doi: 10.1021/acs.orglett.4c03972. Epub 2024 Nov 26.

Abstract

Herein is described the first synthesis of SF5-ynamides, versatile building blocks featuring the pentafluorosulfanyl motif. This synthesis proceeds through a two-step sequence of radical SF5-addition onto the π-system of a wide range of terminal ynamides and derivatives substituted with various nitrogen fragments followed by a dehydrochlorination reaction. A selection of downstream functionalization reactions, including nucleophilic additions, cycloadditions, and sulfur ylide synthesis, highlights the wide-ranging applications of this novel type of functionalized SF5-building block.