Endocannabinoid System and Metabolism: The Influences of Sex

Int J Mol Sci. 2024 Nov 6;25(22):11909. doi: 10.3390/ijms252211909.

Abstract

The endocannabinoid system (ECS) is a lipid signaling system involved in numerous physiological processes, such as endocrine homeostasis, appetite control, energy balance, and metabolism. The ECS comprises endocannabinoids, their cognate receptors, and the enzymatic machinery that tightly regulates their levels within tissues. This system has been identified in various organs, including the brain and liver, in multiple mammalian and non-mammalian species. However, information regarding the sex-specific regulation of the ECS remains limited, even though increasing evidence suggests that interactions between sex steroid hormones and the ECS may ultimately modulate hepatic metabolism and energy homeostasis. Within this framework, we will review the sexual dimorphism of the ECS in various animal models, providing evidence of the crosstalk between endocannabinoids and sex hormones via different metabolic pathways. Additionally, we will underscore the importance of understanding how endocrine-disrupting chemicals and exogenous cannabinoids influence ECS-dependent metabolic pathways in a sex-specific manner.

Keywords: CB1; appetite; endocannabinoid system; lipid signaling; liver; metabolic disorders; sex hormones; sexual dimorphism.

Publication types

  • Review

MeSH terms

  • Animals
  • Brain / metabolism
  • Endocannabinoids* / metabolism
  • Energy Metabolism
  • Female
  • Gonadal Steroid Hormones* / metabolism
  • Humans
  • Liver / metabolism
  • Male
  • Receptors, Cannabinoid / metabolism
  • Sex Characteristics*
  • Signal Transduction

Substances

  • Endocannabinoids
  • Gonadal Steroid Hormones
  • Receptors, Cannabinoid

Grants and funding

M.L. is supported by a postdoctoral contract (Ayudas Margarita Salas para la formación de jóvenes doctores, convocatoria de la Universidad de León de Ayudas para la recualificación del sistema Universitario Español para 2021–2023). F.S. Ph.D. fellowship was founded by UNIVPM.