Her2 promotes early dissemination of breast cancer by inhibiting the p38 pathway through the downregulation of MAP3K4

Cell Commun Signal. 2024 Dec 19;22(1):611. doi: 10.1186/s12964-024-02000-2.

Abstract

Early dissemination refers to the process by which cancer cells spread to distant organs at an early stage of the disease, often before the primary tumor is clinically detectable. Experimental studies have demonstrated that Her2 promotes early dissemination of breast cancer by inhibiting the p38 signaling pathway. However, the precise mechanism by which Her2 suppresses the activation of p38 signaling in early-stage cancer cells (ECCs) remains unclear. Here, we report that MAP3K4, an upstream kinase of p38, is downregulated in Her2 + ductal carcinoma in situ (DCIS) cells and tissues, which is required for Her2-induced early dissemination of DCIS cells by regulating the activation of the p38 signaling cascade. Furthermore, Her2 suppresses the transcription of MAP3K4 by downregulating the expression of HOXB13, a crucial transcription factor contributing to MAP3K4 expression in DCIS cells. Together, these findings unveil a novel downstream regulatory mechanism through which Her2 inhibits the activation of p38 signaling and facilitates early dissemination of breast cancer, offering insights into the development of effective diagnostic methods and targeted therapies for inhibiting the early dissemination of Her2 + breast cancer.

Keywords: Breast cancer; Early dissemination; HOXB13; Her2; MAP3K4; p38.

MeSH terms

  • Animals
  • Breast Neoplasms* / genetics
  • Breast Neoplasms* / metabolism
  • Breast Neoplasms* / pathology
  • Carcinoma, Intraductal, Noninfiltrating / genetics
  • Carcinoma, Intraductal, Noninfiltrating / metabolism
  • Carcinoma, Intraductal, Noninfiltrating / pathology
  • Cell Line, Tumor
  • Down-Regulation*
  • Female
  • Gene Expression Regulation, Neoplastic
  • Homeodomain Proteins / genetics
  • Homeodomain Proteins / metabolism
  • Humans
  • MAP Kinase Kinase Kinase 4 / genetics
  • MAP Kinase Kinase Kinase 4 / metabolism
  • MAP Kinase Signaling System / genetics
  • Mice
  • Receptor, ErbB-2* / genetics
  • Receptor, ErbB-2* / metabolism
  • Signal Transduction
  • p38 Mitogen-Activated Protein Kinases* / metabolism

Substances

  • Receptor, ErbB-2
  • p38 Mitogen-Activated Protein Kinases
  • ERBB2 protein, human
  • Homeodomain Proteins
  • MAP Kinase Kinase Kinase 4