Timing of Dose Reductions and Survival Outcomes in Metastatic Breast Cancer Patients Treated with Cyclin-Dependent Kinase 4/6 Inhibitors

Curr Oncol. 2024 Nov 22;31(12):7426-7436. doi: 10.3390/curroncol31120548.

Abstract

Background/objectives: Dose reductions in CDK4/6 inhibitors, such as ribociclib and palbociclib, are often necessary due to treatment-related toxicities in patients with advanced breast cancer. This study aims to evaluate the impact of the timing of dose reductions on progression-free survival (PFS) and overall survival (OS) in a real-world cohort.

Methods: This single-center, retrospective study included patients treated with ribociclib or palbociclib between 2019 and 2023 at a cancer center in Turkey. Dose reductions due to drug-related toxicities were recorded, and survival outcomes were analyzed. Patients were categorized based on the timing of dose reductions: within the first 3 months (early) and after 3 months (late).

Results: Among 392 patients (mean age 57.13 years), 16.8% had dose reductions within 3 months, 21.7% had late dose reductions, and 61.5% had no dose reductions. The mPFS was 14.26 months for early dose reductions, 33.12 months for late dose reductions, and 20.6 months for no dose reductions (p < 0.001). The mOS was 37.12 months for early dose reductions, not reached for late dose reductions, and 57.76 months for no dose reductions (p < 0.001). Hematological toxicity, primarily neutropenia, was the most common cause of dose reductions. The ECOG performance status, line of therapy, and CDK4/6 inhibitor type were also significant predictors of PFS and OS.

Conclusions: Early dose reductions in CDK4/6 inhibitors negatively affect PFS and OS, highlighting the importance of maintaining treatment intensity in the first 3 months. However, late dose reductions do not negatively affect progression-free survival (PFS) or overall survival (OS), with late dose reductions associated with better outcomes. Prospective studies in larger patient populations will further clarify our knowledge on this subject.

Keywords: CDK4/6 inhibitors; breast cancer; dose reduction; survival outcomes.

MeSH terms

  • Adult
  • Aged
  • Aminopyridines / therapeutic use
  • Breast Neoplasms* / drug therapy
  • Breast Neoplasms* / mortality
  • Breast Neoplasms* / pathology
  • Cyclin-Dependent Kinase 4* / antagonists & inhibitors
  • Cyclin-Dependent Kinase 6* / antagonists & inhibitors
  • Female
  • Humans
  • Middle Aged
  • Neoplasm Metastasis
  • Piperazines* / therapeutic use
  • Progression-Free Survival
  • Protein Kinase Inhibitors* / therapeutic use
  • Purines* / administration & dosage
  • Purines* / therapeutic use
  • Pyridines* / therapeutic use
  • Retrospective Studies

Substances

  • Cyclin-Dependent Kinase 6
  • Cyclin-Dependent Kinase 4
  • palbociclib
  • ribociclib
  • Piperazines
  • Protein Kinase Inhibitors
  • Purines
  • Pyridines
  • Aminopyridines
  • CDK6 protein, human

Grants and funding

This research received no external funding.