SPDEF ameliorates UUO-induced renal fibrosis by transcriptional activation of NR4A1

Mol Med. 2024 Dec 30;30(1):282. doi: 10.1186/s10020-024-01030-3.

Abstract

Nuclear receptor 4A1 (NR4A1) is a gene that increases the likelihood of chronic kidney disease (CKD) and contributes to its development. Previous research has shown that the SAM pointed domain containing Ets transformation-specific transcription factor (SPDEF) can activate NR4A1, but its mechanism of action in renal fibrosis is not yet clear. In this study, we used adenovirus to create a mouse kidney model with a specific knockdown of NR4A1 gene. Our results showed that the knockdown of NR4A1 can accelerate unilateral ureteral obstruction (UUO)-induced renal fibrosis in mice, and overexpression of NR4A1 can significantly reduce transforming growth factor-β1-induced (TGF-β1) fibrosis in HK-2 cells. Additionally, we found that overexpression of SPDEF can improve UUO-induced renal fibrosis in mice and TGF-β1-induced fibrosis in HK-2 by transcriptionally activating NR4A1. These findings suggest that SPDEF can activate NR4A1 transcriptionally and improve renal fibrosis.

Keywords: Chronic kidney disease; NR4A1; Renal fibrosis; SPDEF.

MeSH terms

  • Animals
  • Cell Line
  • Disease Models, Animal*
  • Fibrosis*
  • Gene Knockdown Techniques
  • Humans
  • Kidney / metabolism
  • Kidney / pathology
  • Kidney Diseases / etiology
  • Kidney Diseases / genetics
  • Kidney Diseases / metabolism
  • Kidney Diseases / pathology
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Nuclear Receptor Subfamily 4, Group A, Member 1* / genetics
  • Nuclear Receptor Subfamily 4, Group A, Member 1* / metabolism
  • Proto-Oncogene Proteins c-ets / genetics
  • Proto-Oncogene Proteins c-ets / metabolism
  • Transcriptional Activation*
  • Transforming Growth Factor beta1 / genetics
  • Transforming Growth Factor beta1 / metabolism
  • Ureteral Obstruction* / complications
  • Ureteral Obstruction* / genetics
  • Ureteral Obstruction* / metabolism
  • Ureteral Obstruction* / pathology

Substances

  • Nuclear Receptor Subfamily 4, Group A, Member 1
  • Nr4a1 protein, mouse
  • Transforming Growth Factor beta1
  • Proto-Oncogene Proteins c-ets
  • NR4A1 protein, human