Targeted Activation of OGG1 Inhibits Paraptosis in Lens Epithelial Cells of Early Age-Related Cortical Cataract

Invest Ophthalmol Vis Sci. 2025 Jan 2;66(1):29. doi: 10.1167/iovs.66.1.29.

Abstract

Purpose: To investigate potential modes of programmed cell death in the lens epithelial cells (LECs) of patients with early age-related cortical cataract (ARCC) and to explore early-stage intervention strategies.

Methods: Anterior lens capsules were collected from early ARCC patients for comprehensive analysis. Ultrastructural examination of LECs was performed using transmission electron microscopy. Cell death-associated protein markers were quantified via Western blot analysis, including those for paraptosis (ALIX, GRP78), apoptosis (cleaved caspase 3 and caspase 9), pyroptosis (N-GSDMD), and ferroptosis (GPX4). Intracellular vesicle-organelle colocalization was assessed through immunofluorescence. OGG1 protein expression and activity were evaluated through multiple methods, including Western blot, laser micro-irradiation, and immunofluorescence. The therapeutic potential of the OGG1 activator TH10785 on paraptosis was investigated using an ex vivo rat lens model.

Results: Morphologic changes revealed significant endoplasmic reticulum (ER) swelling in ARCC patient LECs, with no characteristic apoptotic features. Paraptosis-related proteins exhibited significant alterations, while other cell death pathway markers (apoptosis, pyroptosis, and ferroptosis) remained unchanged. In the reactive oxygen species-induced paraptosis model, vesicular structures showed exclusive colocalization with ER-specific fluorescence. Elevated levels of the DNA damage marker 7,8-dihydro-8-oxoguanine were observed concurrent with decreased OGG1 activity. The OGG1 activator TH10785 showed efficacy in suppressing LECs paraptosis in ex vivo rat lens cultures.

Conclusions: Paraptosis was identified in the LECs of patients with early ARCC. TH10785 activates OGG1 to suppress paraptosis in LECs, suggesting a novel therapeutic approach for early ARCC intervention.

MeSH terms

  • Aged
  • Animals
  • Apoptosis / drug effects
  • Blotting, Western
  • Cataract* / metabolism
  • Cataract* / pathology
  • DNA Glycosylases* / metabolism
  • Endoplasmic Reticulum Chaperone BiP
  • Epithelial Cells* / metabolism
  • Female
  • Ferroptosis / drug effects
  • Ferroptosis / physiology
  • Humans
  • Lens, Crystalline / drug effects
  • Lens, Crystalline / metabolism
  • Male
  • Microscopy, Electron, Transmission
  • Middle Aged
  • Paraptosis
  • Pyroptosis / drug effects
  • Rats
  • Rats, Sprague-Dawley

Substances

  • DNA Glycosylases
  • oxoguanine glycosylase 1, human
  • OGG1 protein, rat
  • Endoplasmic Reticulum Chaperone BiP