Gastroprotective effect of fucoidan from Sargassum siliquastrum against ethanol-induced gastric mucosal injury

Food Res Int. 2025 Feb:201:115566. doi: 10.1016/j.foodres.2024.115566. Epub 2024 Dec 30.

Abstract

The ethanol-induced BALB/c mice and human gastric epithelial cell (Ges-1 cell) models were used to investigate the Sargassum siliquastrum fucoidan (SFuc) gastroprotective capability. The injury score and histopathological sections of the stomach were used to evaluate the gastroprotective capability. The western blotting and RT-PCR methods determined the signaling mechanism of mice's gastric injury. SFuc is fucoidan with a molecular weight of 300.7 and 25.1 kDa. The injury score and ulcer index of the SFuc-200 group decreased by 3.85 and 2.06 folds in contrast with the Model group, respectively. The findings indicated that SFuc reduced oxidative stress and inflammatory factor expression in the gastric mucosa by downregulating the levels of associated genes within the TLR-4, MyD88, and MAPK/NF-κB signaling pathways. Meanwhile, the SFuc-200 group promoted the expressions of EGF and PGE 2 by 1.53 and 1.52 folds, respectively. Together with the expression inhibition of p38, ERK, JNK, and NF-κB proteins in gastric tissue to help for differentiation of gastric cells. In addition, SFuc significantly reduced apoptosis occurrence in mice and Ges-1 cells. Our study provides potential mechanism clues of the SFuc's resistance to ethanol-induced gastric mucosal damage, suggesting its potential functional food for gastric protection.

Keywords: Fucoidan; Gastroprotective activity; Ges-1 cell.

MeSH terms

  • Animals
  • Anti-Ulcer Agents / isolation & purification
  • Anti-Ulcer Agents / pharmacology
  • Cell Line
  • Dinoprostone / metabolism
  • Epidermal Growth Factor / metabolism
  • Epithelial Cells / drug effects
  • Epithelial Cells / metabolism
  • Ethanol* / chemistry
  • Gastric Mucosa* / drug effects
  • Gastric Mucosa* / metabolism
  • Gastric Mucosa* / pathology
  • Humans
  • Male
  • Mice
  • Mice, Inbred BALB C*
  • Myeloid Differentiation Factor 88 / metabolism
  • NF-kappa B / metabolism
  • Oxidative Stress* / drug effects
  • Polysaccharides* / chemistry
  • Polysaccharides* / pharmacology
  • Sargassum* / chemistry
  • Signal Transduction / drug effects
  • Stomach Ulcer* / chemically induced
  • Stomach Ulcer* / drug therapy
  • Stomach Ulcer* / prevention & control
  • Toll-Like Receptor 4 / metabolism

Substances

  • fucoidan
  • Ethanol
  • Polysaccharides
  • NF-kappa B
  • Toll-Like Receptor 4
  • Myeloid Differentiation Factor 88
  • Epidermal Growth Factor
  • Anti-Ulcer Agents
  • Dinoprostone
  • Tlr4 protein, mouse