Recent advances on endogenous Na+,K+-ATPase inhibitors: clinical investigation and purification

Clin Exp Hypertens A. 1985;7(5-6):663-72. doi: 10.3109/10641968509077219.

Abstract

Evidence exists which demonstrates the relationship between a Natriuretic Factor or Na+,K+-ATPase inhibitor and volemic expansion, both in man and animal. Patients having extracellular volume expansion have been studied for the effect of their plasma on erythrocytes 3H-ouabain binding. High levels of ouabain-like activity was found in plasma from acromegalic patients and patients with chronic renal failure. High levels were also observed in some hypertensive patients. A partial purification of such a compound was performed from urine of hypertensives. The partially purified compound inhibited to a greater extent the Na+,K+-ATPase semi-purified from dog kidney than that from sheep brain. The present data are consistent with the possible regulation of the activity or the secretion of plasma ouabain-like activity by extracellular volume.

MeSH terms

  • ATPase Inhibitory Protein
  • Acromegaly / blood
  • Animals
  • Binding Sites
  • Brain / enzymology
  • Digitalis / metabolism
  • Dogs
  • Dose-Response Relationship, Drug
  • Erythrocytes / metabolism
  • Humans
  • Hypertension / blood
  • Kidney / enzymology
  • Kidney Failure, Chronic / blood
  • Kinetics
  • Ouabain / blood
  • Plants, Medicinal
  • Plants, Toxic
  • Proteins / isolation & purification*
  • Proteins / metabolism
  • Swine

Substances

  • Proteins
  • Ouabain