Interaction between yeast cytochrome P-450 and chemical carcinogens

Carcinogenesis. 1985 Sep;6(9):1321-5. doi: 10.1093/carcin/6.9.1321.

Abstract

The binding of various chemical carcinogens to the glucose-inducible form of cytochrome (cyt.) P-450 in Saccharomyces cerevisiae was examined with reference to known metabolism in mammalian systems. All the carcinogens examined gave spectral interactions with the yeast cytochrome. The carcinogens benzo[a]pyrene and cyclophosphamide gave Type I binding, while benzidine and 2-naphthylamine gave Type II binding spectra indicating binding at the haem group. Dimethylnitrosamine gave undetectable binding in yeast microsomal fractions, but a Type I binding spectrum was seen with purified cyt. P-450 preparations. The demonstration that these carcinogens bind to yeast cyt. P-450 is discussed in the light of their genotoxicity.

MeSH terms

  • 2-Naphthylamine / metabolism
  • Benzidines / metabolism
  • Benzo(a)pyrene / metabolism
  • Carcinogens / metabolism*
  • Cyclophosphamide / metabolism
  • Cytochrome P-450 Enzyme System / metabolism*
  • Kinetics
  • Microsomes / metabolism
  • Yeasts / metabolism*

Substances

  • Benzidines
  • Carcinogens
  • benzidine
  • Benzo(a)pyrene
  • Cyclophosphamide
  • Cytochrome P-450 Enzyme System
  • 2-Naphthylamine