Phosphorylation and activation of calmodulin-sensitive cyclic nucleotide phosphodiesterase by a brain Ca2+, calmodulin-dependent protein kinase

Life Sci. 1984 Jul 30;35(5):493-9. doi: 10.1016/0024-3205(84)90242-x.

Abstract

A Ca2+, calmodulin-dependent protein kinase from rat brain with a MW of 640,000 phosphorylated calmodulin-sensitive phosphodiesterase from the brain cytosol. The Km of the enzyme for the phosphodiesterase was 5.0 microM and the Vmax was 212 nmol/mg/min. The amount of phosphate incorporated into the phosphodiesterase was 0.7 mol/mol subunit. Phosphorylation of the phosphodiesterase enhanced the enzyme activity by about 20% for hydrolysis of a higher concentration of cyclic AMP.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3',5'-Cyclic-AMP Phosphodiesterases / metabolism*
  • Animals
  • Brain / enzymology*
  • Calmodulin / physiology
  • Cyclic Nucleotide Phosphodiesterases, Type 1
  • Cytosol / enzymology
  • Enzyme Activation
  • Kinetics
  • Molecular Weight
  • Phosphorylation
  • Protein Kinases / metabolism*
  • Rats

Substances

  • Calmodulin
  • Protein Kinases
  • 3',5'-Cyclic-AMP Phosphodiesterases
  • Cyclic Nucleotide Phosphodiesterases, Type 1