A novel non-adrenergic, non-cholinergic nerve-mediated relaxation of the pig bladder neck: an examination of possible neurotransmitter candidates

Eur J Pharmacol. 1984 Apr 6;99(4):287-93. doi: 10.1016/0014-2999(84)90135-3.

Abstract

Electrical field stimulation of the isolated pig bladder neck preparation initiated rapid non-adrenergic, non-cholinergic nerve-mediated relaxations. A wide range of substances were examined as possible candidates for the neurotransmitter involved. Of these, only 5-hydroxytryptamine, vasoactive intestinal polypeptide, adenosine and adenosine 5'-triphosphate produced relaxations. Noradrenaline, acetylcholine, substance P, bradykinin and angiotensin II caused contraction, while neurotensin, somatostatin, bombesin and gamma-amino butyric acid were without effect. The nerve response was not blocked by methysergide, ketanserin, chymotrypsin, apamin or 8-phenyltheophylline, although methysergide antagonised the responses to 5-hydroxytryptamine, chymotrypsin blocked the responses to VIP, and 8-phenyltheophylline antagonised the responses to adenosine and ATP.

MeSH terms

  • Adenosine / physiology
  • Adenosine Triphosphate / physiology
  • Animals
  • Electric Stimulation
  • Female
  • In Vitro Techniques
  • Muscle Relaxation / drug effects
  • Neurotransmitter Agents / physiology*
  • Serotonin / physiology
  • Swine
  • Urinary Bladder / drug effects
  • Urinary Bladder / innervation*
  • Vasoactive Intestinal Peptide / physiology

Substances

  • Neurotransmitter Agents
  • Serotonin
  • Vasoactive Intestinal Peptide
  • Adenosine Triphosphate
  • Adenosine