Studies in radiosensitizing effects of misonidazole and SR-2508 on C3H/He mouse mammary tumors

Radiat Med. 1984 Jan-Mar;2(1):71-5.

Abstract

The radiosensitizing efficacy of SR-2508, a new 2-nitroimidazole, which is less neurotoxic than misonidazole (MISO) was studied using transplantable mammary carcinoma of C3H/He mice. Tumor responses to treatments were evaluated by growth-delay time assay. In single irradiations, the enhancement ratios of 0.5 mmole/kg of MISO and 1.5 mmole/kg of SR-2508, which were equitoxic to C3H/He mice, were 1.42 and 1.84 respectively. In fractionated irradiations with three fractions over two days or five fractions over four days, the enhancement ratios of 1.5 mmole/kg of SR-2508 were 1.40 and 1.34 respectively. On the other hand the enhancement ratios of MISO at the above mentioned dose in respective fractionated irradiations were 1.15 or 1.11. SR-2508 is considered promising as a hypoxic cell radiosensitizer for clinical use.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Etanidazole
  • Female
  • Mammary Neoplasms, Experimental / radiotherapy*
  • Mice
  • Mice, Inbred C3H
  • Misonidazole / therapeutic use*
  • Neoplasm Transplantation
  • Nitroimidazoles / therapeutic use*
  • Radiation-Sensitizing Agents
  • Radiotherapy Dosage
  • Radiotherapy, High-Energy

Substances

  • Nitroimidazoles
  • Radiation-Sensitizing Agents
  • Etanidazole
  • Misonidazole