Calmodulin activates prokaryotic adenylate cyclase

Proc Natl Acad Sci U S A. 1980 Jul;77(7):3841-4. doi: 10.1073/pnas.77.7.3841.

Abstract

The adenylate cyclase of Bordetella pertussis is stimulated 100- to 1000-fold in a dose-dependent manner by calf brain calmodulin. The system has the following properties. (i) The activation is prevented by ethylene glycol bis(beta-aminoethyl ether)-N,N,N',N'-tetraacetic acid and restored by Ca2+. (ii) Oxidation of the methionine residues of calmodulin abolishes the ability to activate the cyclase. (iii) Trifluoperazine inhibits calmodulin-activated cyclase. (iv) A troponin C preparation stimulates the B. pertussis cyclase with < 0.01 the potency of calmodulin. Although calmodulin has not been demonstrated in prokaryotes, this is an example of a (eukaryotic) calmodulin effect in a prokaryote.

MeSH terms

  • Adenylyl Cyclases / metabolism*
  • Bordetella pertussis / enzymology*
  • Calcium / metabolism
  • Calcium-Binding Proteins / pharmacology*
  • Calmodulin / antagonists & inhibitors
  • Calmodulin / pharmacology*
  • Egtazic Acid / pharmacology
  • Enzyme Activation / drug effects
  • Troponin / pharmacology

Substances

  • Calcium-Binding Proteins
  • Calmodulin
  • Troponin
  • Egtazic Acid
  • Adenylyl Cyclases
  • Calcium