Synthesis of N-(2-hydroxypropyl)methacrylamide copolymers with antimicrobial activity

Biomaterials. 1983 Jan;4(1):44-8. doi: 10.1016/0142-9612(83)90069-8.

Abstract

Copolymers of N-(2-hydroxypropyl)methacrylamide which contained up to 20 mol % of p-nitrophenyl esters of N-methacryloylated oligopeptides, and of N-methacryloylaminophenoxyacetic acids (o-, m-, p-) have been prepared. The aminolyses of these polymers with tert. butylamine, ampicillin and 6-aminopenicillanic acid were kinetically characterized. Based on these results polymer bound ampicillin and polymer bound 6-aminopenicillanic acid were prepared. These preparations possessed antimicrobial activity; they inhibited the growth of Staphylococcus aureus 209 P.

MeSH terms

  • Acrylates / chemical synthesis*
  • Ampicillin
  • Anti-Bacterial Agents / chemical synthesis*
  • Anti-Bacterial Agents / pharmacology
  • Bacteria / drug effects
  • Kinetics
  • Methacrylates / chemical synthesis*
  • Methacrylates / pharmacology
  • Penicillanic Acid

Substances

  • Acrylates
  • Anti-Bacterial Agents
  • Methacrylates
  • Ampicillin
  • Penicillanic Acid
  • aminopenicillanic acid
  • 2-hydroxypropyl methacrylate