Effects of calcium on the chick oviduct progesterone receptor

J Steroid Biochem. 1984 Jan;20(1):429-32. doi: 10.1016/0022-4731(84)90247-4.

Abstract

The chick oviduct cytosol progesterone receptor can be transformed to a small form (Rs = 21A, S20,w:2.9) denoted "mero-receptor" by incubation in the presence of Ca2+ [8]. In the molybdate-free cytosol all the progestin binding components could be completely transformed to mero-form by 1 h treatment with 100 mM Ca2+ at 0 degrees C. If EDTA was secondarily added, the ligand was rapidly released. If molybdate (20 mM) containing cytosol was incubated with Ca2+, no radioactivity was found in the meroposition on the Agarose A 0.5 m column, but the bound steroid sedimented at 2.9 S in sucrose gradients containing Ca2+ (and no molybdate). When 20 nM molybdate was added to cytosol containing receptor activated by 0.3 M KCl, complete mero-transformation by Ca2+ was obtained also by the gel filtration criterion, indicating that molybdate does not inhibit the mero-transforming factor. Ligand-free progesterone receptor could also be completely converted to mero-form by endogenous cytosolic transforming factor and calcium. The transforming factor was completely inactivated, when cytosol was run through Agarose A 0.5 m gel. Mero-transformation was found to be irreversible. The purified progesterone receptor subunit 110 K (B) was partially converted to smaller forms by calcium alone (100 mM, 0 degrees C, 1 h) whereas addition of a small amount of cytosol allowed complete conversion to mero-form.

MeSH terms

  • Animals
  • Calcium / pharmacology*
  • Centrifugation, Density Gradient
  • Chickens
  • Chromatography, Agarose
  • Edetic Acid / pharmacology
  • Molybdenum / pharmacology
  • Oviducts / drug effects*
  • Oviducts / metabolism
  • Receptors, Progesterone / drug effects*
  • Receptors, Progesterone / metabolism

Substances

  • Receptors, Progesterone
  • Molybdenum
  • Edetic Acid
  • Calcium