Resistance to 6-thioguanine in spontaneously cycling and in mitogen-stimulated human peripheral lymphocytes

Mutat Res. 1984 Jan;139(1):41-4. doi: 10.1016/0165-7992(84)90120-9.

Abstract

Spontaneously cycling lymphocytes (in cell division in cultures without addition of phytohemagglutinin, PHA) go through the various phases of the first division with the same kinetics as PHA-stimulated cells. In samples from 10 referents, the frequency of spontaneously cycling lymphocytes varied from 8.9 X 10(-5)-9.5 X 10(-3) as indicated with autoradiography on cells in (S + G2) phase determined by flow sorting. In PHA-stimulated samples from the same persons the frequency of 6-thioguanine (TG)-resistant variants was between 4 X 10(-7) and 2.6 X 10(-6), which indicates that most of the spontaneously cycling cells were TG-sensitive. With lymphocytes from one of the referents it was found that: (i) in the presence of 2 X 10(-4) M TG, more than 97% of the spontaneously cycling cells were inhibited before or in early S phase, and (ii) when a flow cytometer was set to sort out TG-resistant cells in late S + G2 phase after 48 h incubation in medium with PHA, the contribution of TG-resistant cells from the spontaneously cycling fraction amounted to less than 2% of the total number of resistant cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Cycle / drug effects
  • Cells, Cultured
  • Drug Resistance
  • Humans
  • Lymphocyte Activation / drug effects
  • Lymphocytes / drug effects
  • Lymphocytes / physiology*
  • Phytohemagglutinins
  • Thioguanine / toxicity*

Substances

  • Phytohemagglutinins
  • Thioguanine