Distinctive biochemical pattern associated with resistance of hepatocytes in hepatocyte nodules during liver carcinogenesis

Environ Health Perspect. 1983 Mar:49:171-4. doi: 10.1289/ehp.8349171.

Abstract

Hepatocyte ("hyperplastic") nodules induced in the liver by initiation with diethylnitrosamine and selected by dietary 2-acetylaminofluorene plus partial hepatectomy ("resistant hepatocyte model") have a special pattern of biochemical behavior and metabolic activity different than that seen acutely with many xenobiotics including many promoting agents and carcinogens. The nodule cells show a very low uptake of 2-acetylaminofluorene, relative to surrounding and normal liver, low levels of activity in the cytochromes P-450 and aryl hydrocarbon hydroxylase, high levels of activity in gamma-glutamyltransferase, microsomal epoxide hydrolase, soluble glutathione-S-transferase and soluble UDP-glucuronyltransferase (UDP-GT(1)) and elevated levels of glutathione. This metabolic pattern appears to maximize the resistance of the nodules to xenobiotics generally, such as 2-acetylaminofluorene, and thereby may account for the resistant behavior of nodule hepatocytes to the inhibition of cell proliferation and the cytotoxicity by 2-acetylaminofluorene and other carcinogens. The possible importance of this seemingly new metabolic program in carcinogenesis is discussed briefly.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 2-Acetylaminofluorene / pharmacology
  • Animals
  • Carcinogens / pharmacology*
  • Diethylnitrosamine / pharmacology
  • Drug Resistance
  • Liver / metabolism*
  • Liver Neoplasms / chemically induced*
  • Liver Neoplasms / metabolism
  • Male
  • Neoplasms, Experimental / chemically induced
  • Rats
  • Rats, Inbred F344
  • Rats, Inbred Strains

Substances

  • Carcinogens
  • Diethylnitrosamine
  • 2-Acetylaminofluorene