Pancreatic porcine phospholipase A2 catalyzed hydrolysis of phosphatidylcholine in lecithin-bile salt mixed micelles: kinetic studies in a lecithin-sodium cholate system

Arch Biochem Biophys. 1983 Mar;221(2):361-70. doi: 10.1016/0003-9861(83)90155-8.

Abstract

Pancreatic porcine phospholipase A2 catalyzed hydrolysis of phosphatidylcholine in bile salt lecithin mixed micelles has been studied, utilizing a series of assay mixtures for which the micellar size, weight, and composition had been experimentally determined. Under these conditions the enzymatic hydrolysis is dependent on the phosphatidylcholine-to-sodium cholate molar ratio within the mixed micelle rather than the bulk concentration of the phospholipid in the mixture: at 5 mM phosphatidylcholine, variation of the NPC/NNaCh ratio from 0.2 to 2.0 increases the enzymatic activity from 82 to 933 mumol/min/mg protein. The initial rates are linear throughout the entire series of assay mixtures, the activity vs micellar concentration curves exhibit saturation behavior, and treatment of the data according to the "surface-as-cofactor" theory provides linear double-reciprocal plots which intersect in one point. The assay system should be applicable for detailed kinetic studies of lipolytic enzymes, including mammalian phospholipases which exhibit rather low activities toward lecithin-Triton X-100 mixed micelles. The system should also provide a convenient basis for mechanistic studies involving the use of inhibitory phospholipid substrate analogs.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Bile Acids and Salts / metabolism*
  • Catalysis
  • Cholic Acid
  • Cholic Acids
  • Elapid Venoms / analysis
  • Hydrolysis
  • Kinetics
  • Micelles
  • Pancreas / enzymology*
  • Phosphatidylcholines / metabolism*
  • Phospholipases / physiology*
  • Phospholipases A / physiology*
  • Phospholipases A2
  • Swine

Substances

  • Bile Acids and Salts
  • Cholic Acids
  • Elapid Venoms
  • Micelles
  • Phosphatidylcholines
  • Phospholipases
  • Phospholipases A
  • Phospholipases A2
  • Cholic Acid