Kinetic analysis of L-lactate transport in human erythrocytes via the monocarboxylate-specific carrier system

Biochim Biophys Acta. 1983 Aug 10;732(3):562-8. doi: 10.1016/0005-2736(83)90232-8.

Abstract

Three parallel pathways of L-lactate transport across the membrane of human red blood cells can be discriminated: (a) by nonionic diffusion; (b) via the band 3 anion exchange protein; and (c) via a specific monocarboxylate carrier system. Influx of lactate via the latter system leads to alkalinization of the medium, suggesting lactate-proton symport. Kinetic analysis of initial lactate influx via the monocarboxylate carrier indicates a symport system with ordered binding of the two ligands, in the sense that a proton binds first to the translocator, followed by lactate binding to the protonated carrier. The influence of varying trans-pH under conditions of net (zero-trans) flux with constant cis-pH indicates that the monocarboxylate translocator should be considered as a mobile carrier, with the ligand-binding sites exposed alternatively to the outside and the inside of the membrane.

MeSH terms

  • Biological Transport, Active
  • Erythrocyte Membrane / metabolism*
  • Erythrocytes / metabolism*
  • Humans
  • Hydrogen-Ion Concentration
  • Kinetics
  • Lactates / blood*
  • Lactic Acid
  • Mathematics
  • Models, Biological

Substances

  • Lactates
  • Lactic Acid