Intraperitoneal cisplatin with systemic thiosulfate protection

Ann Intern Med. 1982 Dec;97(6):845-51. doi: 10.7326/0003-4819-97-6-845.

Abstract

Seventeen patients with intraperitoneal tumors were treated by 4-hour intraperitoneal dialysis with cisplatin alone, or in combination with an intravenous neutralizing agent, sodium thiosulfate. Cisplatin alone, 90 mg/m2 body surface area intraperitoneally, produced nephrotoxicity. When intraperitoneal cisplatin therapy was combined with intravenous thiosulfate treatment, the dose of cisplatin could be escalated to 270 mg/m2 body surface area without causing an increase in serum creatinine levels or undue myelosuppression. Even at doses up to 270 mg/m2, no local toxicity occurred. The peak peritoneal concentration of free reactive cisplatin averaged 21-fold higher than the plasma level, and the area under the peritoneal cisplatin elimination curve averaged 12-fold more than the area under the plasma curve. Neither of these ratios varied significantly with cisplatin dose. Regression of intraperitoneal tumor masses was observed in patients with far-advanced ovarian carcinoma, mesothelioma, and malignant carcinoid.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adult
  • Aged
  • Ascites / drug therapy
  • Cisplatin / administration & dosage*
  • Cisplatin / adverse effects
  • Cisplatin / metabolism
  • Drug Therapy, Combination
  • Female
  • Humans
  • Kinetics
  • Male
  • Middle Aged
  • Peritoneal Dialysis
  • Peritoneal Neoplasms / drug therapy*
  • Thiosulfates / administration & dosage*

Substances

  • Thiosulfates
  • sodium thiosulfate
  • Cisplatin