Synthesis and pharmacological activity of some 2,3-dihydrofuran-2,3-dione derivatives

Pol J Pharmacol Pharm. 1982 Nov-Dec;34(5-6):391-8.

Abstract

New 2,3-dihydrofuran-2,3-dione derivatives (1-11) were obtained by condensation of oxalyl chloride with Schiff bases of acetyl- or benzoylacetone and aromatic amines. These compounds showed only weak sedative action and weak analgesic effect.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 5-Hydroxytryptophan / pharmacology
  • Analgesics / chemical synthesis
  • Animals
  • Anticonvulsants
  • Chemical Phenomena
  • Chemistry
  • Furans / chemical synthesis*
  • Furans / pharmacology
  • Hexobarbital / pharmacology
  • Lethal Dose 50
  • Male
  • Mice
  • Motor Activity / drug effects
  • Sleep / drug effects
  • Time Factors

Substances

  • Analgesics
  • Anticonvulsants
  • Furans
  • Hexobarbital
  • 5-Hydroxytryptophan