Rectal absorption of diazepam in epileptic children

Arch Dis Child. 1982 Apr;57(4):264-7. doi: 10.1136/adc.57.4.264.

Abstract

The absorption of diazepam after rectal administration was studied in children with epilepsy. When given as a solution, diazepam was rapidly absorbed and produced serum diazepam concentrations above 200 ng/ml within 10 minutes in most children. However, a commercial suppository formulation was absorbed slowly and cannot be recommended for urgent treatment of fits. There is a need in the UK for a rapidly absorbed preparation of diazepam which is approved for rectal use.

Publication types

  • Comparative Study

MeSH terms

  • Adolescent
  • Child
  • Child, Preschool
  • Diazepam / administration & dosage
  • Diazepam / metabolism*
  • Epilepsy / drug therapy
  • Epilepsy / metabolism*
  • Humans
  • Infant
  • Intestinal Absorption*
  • Rectum / metabolism*
  • Solutions
  • Suppositories
  • Time Factors

Substances

  • Solutions
  • Suppositories
  • Diazepam