Inhibition of mutagenesis in Chinese hamster V-79 cells by antioxidants

Toxicol Lett. 1980 Dec;7(2):125-30. doi: 10.1016/0378-4274(80)90044-2.

Abstract

The mutagenicity of benzo(a)pyrene (BP) on Chinese hamster V-79 cells cocultivated with X-irradiated hamster embryo cells was inhibited by phenolic antioxidants, such as tert-butyl-4-hydroxyanisole (BHA) and butyl-hydroxytoluene (BHT), but not by disulfiram and its related compounds such as tetraethylthiuram disulfide, diethyldithiocarbamic acid and dimethyldithiocarbamic acid. The mutagenicity of BP on V-79 cells was reduced 44% by BHA and 25% by BHT. BHA inhibited BP-induced mutagenesis, but not N-acetoxy-2-acetylaminofluorene (N-acetoxy-AAF)-induced mutagenesis. BHA is suggested to inhibit the mutagenic action of BP by altering its metabolism.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / pharmacology*
  • Benzopyrenes / antagonists & inhibitors
  • Biotransformation
  • Cricetinae
  • Cricetulus
  • Mutagens* / metabolism
  • Mutation
  • Phenols / pharmacology

Substances

  • Antioxidants
  • Benzopyrenes
  • Mutagens
  • Phenols