Synthesis of steroidal 17 beta-carboxamide derivatives

Steroids. 1980 Mar;35(3):265-71. doi: 10.1016/0039-128x(80)90039-2.

Abstract

Several 17 beta-carboxamide derivatives of natural and fluorinated glucocorticoids have been synthesized. The 17 beta-carboxylic derivatives were obtained by periodic acid oxidation of their side chains. They were then activated by N-hydroxybenzotriazole (HOBT) and coupled to several primary amines. Using this method eleven 17 beta-carboxamide derivatives have been prepared in good yields.

MeSH terms

  • Chemical Phenomena
  • Chemistry
  • Corticosterone / analogs & derivatives
  • Desoximetasone / analogs & derivatives
  • Dexamethasone / analogs & derivatives
  • Glucocorticoids / chemical synthesis*
  • Hydrocortisone / analogs & derivatives
  • Methods

Substances

  • Glucocorticoids
  • Desoximetasone
  • Dexamethasone
  • Corticosterone
  • Hydrocortisone