Anti-inflammatory activity of croconazole, a broad-spectrum antimycotic agent, in the arachidonic acid-induced mouse ear swelling test

Skin Pharmacol. 1995;8(4):211-4. doi: 10.1159/000211349.

Abstract

Investigations on croconazole, a novel imidazole compound, suggested antiphlogistic properties in vitro. Hence, its anti-inflammatory capacity was tested in vivo using the arachidonic acid-induced mouse ear swelling test, which is a suitable model for screening inhibitors of the lipoxygenase and/or the cyclooxygenase. Topical application of croconazole (1%/0.01%) to the mouse ear induced a maximal inhibition of edema (inhibition: 39%/33%; p = 0.01) which was as strong as the reference nordihydroguaiaretic acid (inhibition: 38.9%; p = 0.01). These results justify further investigations on croconazole to study potential inhibitory effects on proinflammatory arachidonic acid metabolites.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Antifungal Agents / pharmacology*
  • Arachidonic Acid
  • Ear, External / pathology
  • Edema / chemically induced
  • Edema / pathology
  • Edema / prevention & control*
  • Female
  • Guaiacol / analogs & derivatives
  • Guaiacol / pharmacology
  • Imidazoles / pharmacology*
  • Lignans / pharmacology
  • Lipoxygenase Inhibitors / pharmacology
  • Mice
  • Mice, Inbred Strains

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Antifungal Agents
  • Imidazoles
  • Lignans
  • Lipoxygenase Inhibitors
  • Arachidonic Acid
  • dihydroguaiaretic acid
  • croconazole
  • Guaiacol