Mechanisms of the inhibition of reverse transcription by unmodified and modified antisense oligonucleotides

Nucleic Acids Symp Ser. 1993:(29):67-8.

Abstract

We have demonstrated that the synthetic oligonucleotides, either unmodified or phosphorothioates, prevent cDNA synthesis by the AMV or HIV reverse transcriptases. The RNA was truncated at the antisense oligonucleotide-RNA duplex during the reverse transcription. Th blockage involves the degradation of the RNA fragment bound to the antisense oligonucleotide by the reverse transcriptase associated RNase H activity. However, in the case of phosphorothioate oligomer, the production of cDNA would be inhibited by a hybrid formed between the AMV RT and phosphorothioate oligomer than arrested elongation of the cDNA strands, whereas arrest of a growing cDNA strand by HIV RT can be blocked by an oligonucleotide complementary to a region downstream from the primer.

MeSH terms

  • Animals
  • Avian Myeloblastosis Virus / enzymology
  • DNA, Complementary / biosynthesis
  • Globins / genetics
  • HIV / enzymology
  • Oligonucleotides, Antisense / chemistry
  • Oligonucleotides, Antisense / pharmacology*
  • RNA, Messenger / genetics
  • Rabbits
  • Reverse Transcriptase Inhibitors*
  • Thionucleotides / pharmacology
  • Transcription, Genetic / drug effects*

Substances

  • DNA, Complementary
  • Oligonucleotides, Antisense
  • RNA, Messenger
  • Reverse Transcriptase Inhibitors
  • Thionucleotides
  • Globins