A phosphorothioate oligonucleotide blocks reverse transcription via an antisense mechanism

FEBS Lett. 1994 Mar 7;340(3):236-40. doi: 10.1016/0014-5793(94)80145-2.

Abstract

We have studied the inhibition by a phosphorothioate oligodeoxynucleotide (17PScap) of cDNA synthesis performed by either avian or murine reverse transcriptase. Three different mechanisms of inhibition were identified: at low concentrations (< 100 nM), the cleavage of the RNA template by the retroviral RNase H at the level of the RNA/17PScap duplex accounted for most of the effect, whereas hybrid-arrested cDNA synthesis by an RNase H-independent mechanism marginally contributed to the inhibition. Both mechanisms were sequence-specific. Above 100 nM, the overall cDNA synthesis was reduced in a non-specific manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Birds
  • DNA, Complementary / biosynthesis
  • Hydrolysis
  • Mice
  • Molecular Sequence Data
  • Oligonucleotides, Antisense / pharmacology*
  • RNA-Directed DNA Polymerase / metabolism
  • Ribonuclease H / metabolism
  • Templates, Genetic
  • Thionucleotides / pharmacology*
  • Transcription, Genetic / genetics*

Substances

  • DNA, Complementary
  • Oligonucleotides, Antisense
  • Thionucleotides
  • RNA-Directed DNA Polymerase
  • Ribonuclease H