Effect of fepradinol on rat hind paw oedema induced by several inflammatory agents

J Pharm Pharmacol. 1993 Nov;45(11):959-62. doi: 10.1111/j.2042-7158.1993.tb05635.x.

Abstract

Fepradinol is an effective non-steroidal anti-inflammatory agent. The effect on rat paw oedema induced by various phlogistic agents was investigated. The inhibitory effect of fepradinol (25 mg kg-1, p.o.) on dextran-induced oedema was nearly equal to that of cyproheptadine (10 mg kg-1, p.o.). On oedema induced by platelet-activating factor only fepradinol (25 mg kg-1, p.o.) and phenidone (100 mg kg-1, p.o.) clearly inhibited the inflammatory process. Both the above induced oedemas are thought to be unrelated to prostaglandins in the rat system and therefore, the anti-inflammatory activity against them is not shared by selective cyclo-oxygenase inhibitors. Fepradinol (25 mg kg-1, p.o.) displayed an inhibitory effect on the early and late stage of kaolin- and nystatin-induced oedemas in contrast with indomethacin (10 mg kg-1, p.o.) and piroxicam (10 mg kg-1, p.o.) which only inhibited the late stage. The results obtained in this study confirm that fepradinol is a potent anti-inflammatory agent and indicate that its mechanism of action is different from that of other anti-inflammatory compounds.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Dextrans
  • Edema / chemically induced
  • Edema / drug therapy*
  • Edema / pathology
  • Ethanolamines / therapeutic use*
  • Foot / pathology
  • Kaolin
  • Male
  • Nystatin
  • Platelet Activating Factor
  • Rats
  • Rats, Wistar

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Dextrans
  • Ethanolamines
  • Platelet Activating Factor
  • Nystatin
  • Kaolin
  • fepradinol