Mutual inhibition of murine erythropoiesis and granulopoiesis during combined erythropoietin, granulocyte colony-stimulating factor, and stem cell factor administration: in vivo interactions and dose-response surfaces

Blood. 1994 Dec 15;84(12):4157-63.

Abstract

We investigated the in vivo effects of erythropoietin (EPO) on granulopoiesis and, conversely, the effect of granulocyte colony-stimulating factor (G-CSF) treatment on erythropoiesis. Recombinant human EPO at four different doses in combination with recombinant human G-CSF also at four different doses was simultaneously administered for 7 days to splenectomized mice. In total, 16 different combinations of growth factors were thus tested. G-CSF administration increased granulocyte production as expected, whereas immature colony-forming unit granulocyte-macrophage numbers were decreased. EPO analogously increased late erythroid cell numbers. Both EPO and G-CSF dose-dependently inhibited late cell stages of the opposite lineage, with EPO abrogating G-CSF-stimulated granulopoiesis and, conversely, G-CSF inhibiting EPO-stimulated erythropoiesis. In a subsequent experiment, we tested whether these lineage-competitive effects could be prevented by coadministering stem cell factor (SCF). In these three factor-treated mice, all granuloid and erythroid cell stages increased, thereby reducing the effect of the mutual inhibition. We conclude that EPO-stimulated erythropoiesis and G-CSF-stimulated granulopoiesis inhibited each other at a late level. Simultaneous SCF administration increased the input into both the erythroid and granuloid compartment and thereby compensated the mutual inhibition. This study shows that intricate dose-response relationships exist between various growth factors that should be carefully analyzed before combinations of these factors are used in humans.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Dose-Response Relationship, Drug
  • Drug Antagonism
  • Erythropoiesis / drug effects
  • Erythropoietin / pharmacology*
  • Granulocyte Colony-Stimulating Factor / pharmacology*
  • Granulocytes*
  • Hematopoiesis / drug effects*
  • Hematopoietic Cell Growth Factors / pharmacology*
  • Mice
  • Mice, Inbred C57BL
  • Recombinant Proteins / pharmacology
  • Regression Analysis
  • Splenectomy
  • Stem Cell Factor

Substances

  • Hematopoietic Cell Growth Factors
  • Recombinant Proteins
  • Stem Cell Factor
  • Erythropoietin
  • Granulocyte Colony-Stimulating Factor