Staurosporine can inhibit the G1-S transition induced by a calcium channel agonist by blocking the pathway independent of phorbol ester-sensitive protein kinase C in rat thyroid cells (FRTL-5)

Endocr Res. 1994 Aug;20(3):235-45. doi: 10.1080/07435809409035861.

Abstract

IGF-I, when added to TSH-primed FRTL-5 cells, can induce a long lasting Ca2+ influx followed by the DNA synthesis. BAY K8644, a Ca2+ channel agonist, can also induce the DNA synthesis in TSH-treated cells. Staurosporine, which is known to be a potent inhibitor of protein kinase C(PKC) strongly inhibited the DNA synthesis caused by these two reagents. However, in PKC-down regulated cells, IGF-I and BAY K8644 could also evoke the DNA synthesis and the inhibitory effect of staurosporine persisted. These inhibitory effects did not relay on inhibition of the Ca2+ influx induced by BAY K8644. Thus these results demonstrate that staurosporine acts at a point distal to Ca2+ influx to inhibit G1-S transition and this staurosporine-sensitive pathway possibly mediates the mitogenic signal in PKC-independent manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester / pharmacology*
  • Alkaloids / pharmacology*
  • Animals
  • Calcium / metabolism
  • Calcium Channels / drug effects
  • Cell Line
  • G1 Phase / drug effects*
  • Protein Kinase C / metabolism
  • Rats
  • S Phase / drug effects*
  • Staurosporine
  • Tetradecanoylphorbol Acetate / pharmacology
  • Thyroid Gland / cytology*
  • Thyroid Gland / enzymology

Substances

  • Alkaloids
  • Calcium Channels
  • 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester
  • Protein Kinase C
  • Staurosporine
  • Tetradecanoylphorbol Acetate
  • Calcium