[Single channel analysis of aconitine blockade of calcium channels in rat myocardiocytes]

Yao Xue Xue Bao. 1995;30(3):168-71.
[Article in Chinese]

Abstract

Ventricular myocardiocytes from neonatal Wistar rats were isolated and cultured. Aconitine, Ca2+ channel blocker verapamil or Ca2+ channel activator BAY K8644 were added to the bath solution separately. Using the cell-attached configuration of the patch clamp technique, the single channel activities of L type Ca2+ channel were recorded before and after addition of all three drugs. The results showed the blocking effect of aconitine (50 micrograms.ml-1) on L type Ca2+ channels. Its mechanism may be relevant to the decrease in both open state probability and the mean open time of Ca2+ channel. The difference was statistically significant compared with control group (P < 0.01). The amplitude of Ba2+ currents, which flow through open L type Ca2+ channel was unchanged.

Publication types

  • Comparative Study
  • English Abstract

MeSH terms

  • 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester / pharmacology
  • Aconitine / pharmacology*
  • Animals
  • Animals, Newborn
  • Calcium Channel Blockers / pharmacology*
  • Cells, Cultured
  • Myocardium / cytology*
  • Rats
  • Rats, Wistar
  • Verapamil / pharmacology

Substances

  • Calcium Channel Blockers
  • 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester
  • Verapamil
  • Aconitine