Activity of ecdysone analogs in enhancing N-acetylglucosamine incorporation into the cultured integument of Chilo suppressalis

Steroids. 1995 May;60(5):401-5. doi: 10.1016/0039-128x(94)00065-k.

Abstract

Ecdysone analogs with various side chains at the 17-position of the steroid structure enhanced the incorporation of N-acetylglucosamine as 20-hydroxyecdysone into the cultured integument prepared from Chilo suppressalis. Their activity in terms of the concentration required to give 50% of the maximum response varied with the structure. Piperonyl butoxide, an inhibitor of oxidation metabolism, did not enhance the in vitro effect of the compounds. The order of potency was ponasterone A > 20-hydroxyecdysone > cyasterone > inokosterone > makisterone A >> ecdysone.

MeSH terms

  • Acetylglucosamine / metabolism*
  • Animals
  • Cells, Cultured
  • Chitin / biosynthesis
  • Cholestanes / chemistry
  • Cholestanes / pharmacology
  • Dose-Response Relationship, Drug
  • Drosophila
  • Ecdysone / analogs & derivatives*
  • Ecdysone / pharmacology*
  • Insect Hormones / chemistry
  • Insect Hormones / pharmacology*
  • Lepidoptera / metabolism*
  • Piperonyl Butoxide / pharmacology
  • Structure-Activity Relationship

Substances

  • Cholestanes
  • Insect Hormones
  • Chitin
  • Ecdysone
  • Piperonyl Butoxide
  • Acetylglucosamine