Acrylic acid oxidation and tissue-to-blood partition coefficients in rat tissues

Toxicol Lett. 1995 Jun;78(1):73-8. doi: 10.1016/0378-4274(94)03233-w.

Abstract

We report rates of acrylic acid (AA) oxidation and tissue/blood partition coefficients in rat tissues. AA oxidation in Fischer 344 rat kidney and liver slices was described by saturable kinetics with maximal velocities of about 4 and 2 mumol/h/g, respectively. AA oxidation rates in 11 additional tissues were 40% or less than in liver. AA oxidation rates in Sprague-Dawley rat liver and kidney were similar to those in Fischer rats. Partition coefficients varied within a narrow range, suggesting that a tissue's contribution to systemic detoxification of AA will depend much more strongly on its rate of AA oxidation and the proportion of the cardiac output that it receives.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrylates / blood
  • Acrylates / pharmacokinetics*
  • Animals
  • Culture Techniques
  • Dose-Response Relationship, Drug
  • Kidney / metabolism*
  • Liver / metabolism*
  • Male
  • Oxidation-Reduction
  • Rats
  • Rats, Inbred F344
  • Rats, Sprague-Dawley
  • Species Specificity
  • Tissue Distribution

Substances

  • Acrylates
  • acrylic acid