Differential effects by Mad and Max on transformation by cellular and viral oncoproteins

Oncogene. 1995 Aug 3;11(3):587-96.

Abstract

c-Myc is an essential component of the regulatory mechanisms controlling cell growth. Max is the obligatory partner of c-Myc for all its biological functions analysed to date. Recently two Max interacting proteins, Mad and Mxi1, have been identified. It has been suggested that these two proteins modulate c-Myc function, in the simplest model by competing with c-Myc for the interaction with Max. We have analysed different aspects of Mad function in comparison to Max. Native Mad/Max heterodimers bound specifically to a c-Myc/Max consensus DNA binding site. Furthermore Mad inhibited efficiently c-Myc, mutant p53, adenovirus E1a, or human papilloma virus type 16 transformation of rat embryo cells in cooperation with activated Ha-Ras. Myc transformed clones showed an increased cell cycle time and a reduced immortalization frequency after cotransfection with either mad or max. In contrast to Mad, Max did not inhibit E1a/Ha-Ras cotransformation but repressed c-Myc/Ha-Ras transformation efficiently. Mad delta N, an N-terminal deletion mutant of Mad, was as efficient in repressing c-Myc/Ha-Ras cotransformation as full length Mad but showed little inhibitory activity when assayed on E1a/Ha-Ras. Unlike wt Mad, Mad delta N had little effect on cell growth. Our data suggest that Mad affects cell growth at least in part by a c-Myc independent mechanism.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Basic Helix-Loop-Helix Leucine Zipper Transcription Factors
  • Basic-Leucine Zipper Transcription Factors
  • Cell Cycle
  • Cell Line
  • Cell Transformation, Neoplastic*
  • Chlorocebus aethiops
  • DNA-Binding Proteins / physiology*
  • Gene Expression
  • Genes, myc
  • Genes, ras
  • Macromolecular Substances
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Oligodeoxyribonucleotides / chemistry
  • Oncogene Proteins, Viral / physiology*
  • Proto-Oncogene Proteins c-myc / physiology*
  • Proto-Oncogene Proteins p21(ras) / physiology*
  • RNA, Messenger / genetics
  • Repressor Proteins*
  • Structure-Activity Relationship
  • Transcription Factors*
  • Transfection

Substances

  • Basic Helix-Loop-Helix Leucine Zipper Transcription Factors
  • Basic-Leucine Zipper Transcription Factors
  • DNA-Binding Proteins
  • MXD1 protein, human
  • Macromolecular Substances
  • Myc associated factor X
  • Oligodeoxyribonucleotides
  • Oncogene Proteins, Viral
  • Proto-Oncogene Proteins c-myc
  • RNA, Messenger
  • Repressor Proteins
  • Transcription Factors
  • Proto-Oncogene Proteins p21(ras)