Analysis of the proenkephalin second messenger-inducible enhancer in rat striatal cultures

J Neurochem. 1995 Sep;65(3):1007-15. doi: 10.1046/j.1471-4159.1995.65031007.x.

Abstract

We have previously shown that in cell extracts from rat striatum, cyclic AMP response element (CRE) binding protein (CREB), rather than AP-1 proteins, preferentially interacts with the CRE-2 element of the proenkephalin second messenger-inducible enhancer, even under conditions in which AP-1 proteins are highly induced. Here we use primary striatal cultures to permit a more detailed analysis of CRE-2 function and protein binding in relevant neural cell types. By transfection we find that in primary striatal cultures, as in transformed cell lines, the CRE-1 and CRE-2 elements are required for significant induction by cyclic AMP. We report that cyclic AMP induction of the proenkephalin gene in striatal cultures is protein synthesis independent, excluding a role for newly synthesized proteins like c-Fos. We also show that cyclic AMP induces CREB phosphorylation and that phosphorylated CREB interacts strongly with CRE-2 and weakly with CRE-1. The predominant protein bound to CRE-1 is not CREB, however, and remains to be identified. Despite some prior predictions, we do not find a role for c-Fos in cyclic AMP regulation of proenkephalin gene expression in neurons.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone / pharmacology
  • Adenosine / analogs & derivatives
  • Adenosine / pharmacology
  • Adenosine-5'-(N-ethylcarboxamide)
  • Animals
  • Base Sequence
  • Cells, Cultured
  • Colforsin / pharmacology
  • Corpus Striatum / metabolism*
  • Cyclic AMP / pharmacology
  • Cyclic AMP Response Element-Binding Protein / metabolism
  • Enhancer Elements, Genetic*
  • Enkephalins / genetics*
  • Fetus
  • Genes, fos
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Precursors / genetics*
  • RNA, Messenger / biosynthesis
  • Rats
  • Rats, Sprague-Dawley
  • Second Messenger Systems*
  • Transcription Factor AP-1 / metabolism

Substances

  • Cyclic AMP Response Element-Binding Protein
  • Enkephalins
  • Protein Precursors
  • RNA, Messenger
  • Transcription Factor AP-1
  • proenkephalin
  • Colforsin
  • 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone
  • Adenosine-5'-(N-ethylcarboxamide)
  • Cyclic AMP
  • Adenosine