Synthesis and antimicrobial evaluation of 4-phenyl-3-isoquinolinoyl-hydrazones

Farmaco. 1995 Apr;50(4):265-72.

Abstract

2-Methyl-1-oxo-1,2-dihydro-3-carbazoyl-4-phenylisoquinoline 2, 1-methoxy-7 and 1-chloro-3-carbazoyl-4-phenylisoquinoline 12 as well as a series of their 2-hydrazono-derivatives 3 a-i, 8 a-i and 14 a-i were synthesized and evaluated for their antibacterial and antifungal activities, in vitro. Compound 3 h was fairly active against Staphylococcus aureus, Staphylococcus epidermidis and streptococci group B.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / chemical synthesis*
  • Anti-Bacterial Agents / pharmacology
  • Gram-Negative Bacteria / drug effects
  • Gram-Positive Bacteria / drug effects
  • Hydrazones / chemical synthesis*
  • Hydrazones / pharmacology
  • Isoquinolines / chemical synthesis*
  • Isoquinolines / pharmacology
  • Molecular Structure

Substances

  • Anti-Bacterial Agents
  • Hydrazones
  • Isoquinolines