Evidence for a membrane exchangeable glucose pool in the functioning of rat liver glucose-6-phosphatase

J Biol Chem. 1995 Sep 8;270(36):21098-102.

Abstract

We have investigated the kinetics of tracer uptake into rat liver microsomes in relation to [14C]glucose 6-phosphate (Glu-6-P) hydrolysis by glucose 6-phosphatase (Glu-6-Pase). 1) The steady-state levels of intravesicular tracer accumulated during the rapid (AMP1) and slow (AMP2) phases of uptake both demonstrate Michaelis-Menten kinetics relative to outside Glu-6-P concentrations with Km values similar to those observed for the initial burst (Vi) and steady-state (VSS) rates of Glu-6-P hydrolysis. 2) The AMP1/AMP2 ratio is constant (mean value = 0.105 +/- 0.018) over the whole range of outside Glu-6-P concentrations and is equal to the AMP1max/AMP2max ratio (0.109 +/- 0.032). 3) Linear relationships are observed between the initial rates of glucose transport during the slow uptake phase (V alpha 2) and [AMP1], and between [VSS] and [AMP2]. 4) The value of Vss max exceeds by more than 10-fold that of V alpha 2 max. 5) It is concluded that the substrate transport model is incompatible with those results and that AMP1 represents a membrane exchangeable glucose pool. 6) We propose a new version of the conformational model in which the catalytic site lies deep within a hydrophilic pocket of an intrinsic membrane protein and communicates with the extra- and intravesicular spaces through channels with different glucose permeabilities.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Membrane / metabolism
  • Cell Membrane Permeability
  • Glucose / metabolism*
  • Glucose-6-Phosphatase / metabolism*
  • Glucose-6-Phosphate
  • Glucosephosphates / metabolism*
  • Hydrolysis
  • Kinetics
  • Male
  • Microsomes, Liver / enzymology
  • Microsomes, Liver / metabolism*
  • Rats
  • Rats, Wistar

Substances

  • Glucosephosphates
  • Glucose-6-Phosphate
  • Glucose-6-Phosphatase
  • Glucose