Effects of dipyridamole and R-verapamil on in vitro proliferation of blast cells from patients with acute myelogenous leukaemia

Leuk Res. 1993 Jun;17(6):507-13. doi: 10.1016/0145-2126(93)90126-6.

Abstract

Cytokine-dependent AML cell proliferation was investigated in 16 patients. Dipyridamole and R-verapamil caused a dose-dependent inhibition of AML cell proliferation, and for both drugs the degree of inhibition was similar when testing various haematopoietic growth factors or growth factor combinations (IL3, G-CSF, GM-CSF, G-CSF + GM-CSF, TNF-alpha + GM-CSF). TNF-alpha alone increased AML cell proliferation for five patients, whereas four patients showed unaltered or decreased proliferation. Independent of this TNF-alpha effect, R-verapamil inhibited proliferation for all AML patients in the presence of TNF-alpha, whereas dipyridamole caused only a weak inhibition.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Blast Crisis / pathology*
  • Cell Division / drug effects*
  • Cell Division / radiation effects
  • Dipyridamole / pharmacology*
  • Dose-Response Relationship, Drug
  • Female
  • Granulocyte Colony-Stimulating Factor / pharmacology
  • Granulocyte-Macrophage Colony-Stimulating Factor / pharmacology
  • Growth Substances / pharmacology*
  • Hematopoietic Cell Growth Factors / pharmacology*
  • Humans
  • Interleukin-3 / pharmacology
  • Kinetics
  • Leukemia, Myeloid, Acute / pathology*
  • Male
  • Middle Aged
  • Recombinant Proteins / pharmacology
  • Tumor Cells, Cultured
  • Tumor Necrosis Factor-alpha / pharmacology
  • Verapamil / pharmacology*

Substances

  • Growth Substances
  • Hematopoietic Cell Growth Factors
  • Interleukin-3
  • Recombinant Proteins
  • Tumor Necrosis Factor-alpha
  • Granulocyte Colony-Stimulating Factor
  • Dipyridamole
  • Granulocyte-Macrophage Colony-Stimulating Factor
  • Verapamil