Involvement of GPIIb-IIIa on human platelets in phosphotyrosine-specific dephosphorylation

Biochem Biophys Res Commun. 1993 Jul 15;194(1):472-7. doi: 10.1006/bbrc.1993.1843.

Abstract

Washed platelets from either normal donors or patients with thrombasthenia lacking in integrin GPIIb-IIIa were stimulated by thrombin or STA2 with stirring and their kinetics of protein-tyrosine phosphorylation were compared. The early increase in protein-tyrosine phosphorylation on 115 and 75 kDa protein bands was observed within 10 s after stimulation in both normal and thrombasthenic platelets. While both 115 and 75 kDa tyrosine-phosphorylated protein bands were quickly dephosphorylated in normal platelets, thrombin-induced 115 kDa or STA2-induced 115 and 75 kDa protein bands were not dephosphorylated in thrombasthenic platelets. The delay of phosphotyrosine-specific dephosphorylation on those protein bands was observed when thrombin- or STA2-induced aggregation of normal platelets was inhibited by RGDS, an inhibitor of fibrinogen binding to GPIIb-IIIa. These data indicate that fibrinogen binding to GPIIb-IIIa is involved in the regulation of phosphotyrosine-specific dephosphorylation on certain protein bands.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Antibodies
  • Antibodies, Monoclonal
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism*
  • Humans
  • Immunoblotting
  • In Vitro Techniques
  • Kinetics
  • Molecular Weight
  • Oligopeptides / metabolism
  • Phosphoproteins / blood*
  • Phosphoproteins / isolation & purification
  • Phosphotyrosine
  • Platelet Membrane Glycoproteins / genetics
  • Platelet Membrane Glycoproteins / metabolism*
  • Reference Values
  • Thrombasthenia / blood*
  • Thrombin / pharmacology
  • Thromboxane A2 / analogs & derivatives
  • Thromboxane A2 / pharmacology
  • Tyrosine / analogs & derivatives*
  • Tyrosine / blood

Substances

  • Antibodies
  • Antibodies, Monoclonal
  • Oligopeptides
  • Phosphoproteins
  • Platelet Membrane Glycoproteins
  • Phosphotyrosine
  • Tyrosine
  • Thromboxane A2
  • STA 2
  • arginyl-glycyl-aspartyl-serine
  • Thrombin