Beta-endorphin binding activity of SP-40,40

Biol Pharm Bull. 1993 Mar;16(3):228-31. doi: 10.1248/bpb.16.228.

Abstract

SP-40,40 bound to beta-endorphin via C-terminal non-opioid portion of beta-endorphin as well as S-protein (vitronectin) bound. Beta-endorphin bound mainly to SP-40,40, but not to S-protein, in the soluble membrane attack complex (SMAC, SC5b-9) of complement, because the results of autoradiography of the cross-linking experiment of SMAC with [125I] beta-endorphin revealed only a typical band of SP-40,40. The binding of SP-40,40 to beta-endorphin inhibited the binding of beta-endorphin to its receptor of rat brain; thus SP-40,40 might inhibit the biological action of beta-endorphin.

MeSH terms

  • Animals
  • Autoradiography
  • Clusterin
  • Complement Membrane Attack Complex / metabolism
  • Cross-Linking Reagents / pharmacology
  • Extracellular Matrix Proteins / metabolism
  • Glycoproteins / metabolism*
  • Glycoproteins / pharmacology
  • Humans
  • In Vitro Techniques
  • Iodine Radioisotopes
  • Molecular Chaperones*
  • Nerve Tissue Proteins / metabolism*
  • Nerve Tissue Proteins / pharmacology
  • Protein Binding
  • Rats
  • Receptors, Opioid / drug effects
  • Receptors, Opioid / metabolism
  • Vitronectin
  • beta-Endorphin / metabolism*

Substances

  • CLU protein, human
  • Clusterin
  • Complement Membrane Attack Complex
  • Cross-Linking Reagents
  • Extracellular Matrix Proteins
  • Glycoproteins
  • Iodine Radioisotopes
  • Molecular Chaperones
  • Nerve Tissue Proteins
  • Receptors, Opioid
  • Vitronectin
  • beta-Endorphin