Functional interactions in bacteriorhodopsin: a theoretical analysis of retinal hydrogen bonding with water

Biophys J. 1995 Jan;68(1):25-39. doi: 10.1016/S0006-3495(95)80184-0.

Abstract

The light-driven proton pump, bacteriorhodopsin (bR) contains a retinal molecule with a Schiff base moiety that can participate in hydrogen-bonding interactions in an internal, water-containing channel. Here we combine quantum chemistry and molecular mechanics techniques to determine the geometries and energetics of retinal Schiff base-water interactions. Ab initio molecular orbital calculations are used to determine potential surfaces for water-Schiff base hydrogen-bonding and to characterize the energetics of rotation of the C-C single bond distal and adjacent to the Schiff base NH group. The ab initio results are combined with semiempirical quantum chemistry calculations to produce a data set used for the parameterization of a molecular mechanics energy function for retinal. Using the molecular mechanics force field the hydrated retinal and associated bR protein environment are energy-minimized and the resulting geometries examined. Two distinct sites are found in which water molecules can have hydrogen-bonding interactions with the Schiff base: one near the NH group of the Schiff base in a polar region directed towards the extracellular side, and the other near a retinal CH group in a relatively nonpolar region, directed towards the cytoplasmic side.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bacteriorhodopsins / chemistry*
  • Binding Sites
  • Biophysical Phenomena
  • Biophysics
  • Crystallography, X-Ray
  • Electrochemistry
  • Halobacterium salinarum / chemistry
  • Hydrogen Bonding
  • Models, Chemical
  • Models, Molecular
  • Protein Conformation
  • Protons
  • Retinaldehyde / chemistry
  • Schiff Bases / chemistry
  • Thermodynamics
  • Water / chemistry

Substances

  • Protons
  • Schiff Bases
  • Water
  • Bacteriorhodopsins
  • Retinaldehyde