Potentiation by tumour necrosis factor-alpha of calcium signals induced by bradykinin and carbachol in human tracheal smooth muscle cells

Br J Pharmacol. 1995 Jan;114(1):4-5. doi: 10.1111/j.1476-5381.1995.tb14896.x.

Abstract

The effect of tumour necrosis factor-alpha (TNF alpha) on the increase in cytosolic free calcium ([Ca2+])i induced by carbachol and bradykinin (BK) was investigated in human tracheal smooth muscle cells in culture (TSMC). BK (10(-12)-10(-9) M) and carbachol (10(-7)-10(-3) M) produced a concentration-dependent increase in [Ca2+]i (pD2 = 10.73 +/- 0.05 and 5.57 +/- 0.03 respectively). The increase in [Ca2+]i was significantly enhanced for both agonists in TNF alpha-treated cells (10 ng ml-1 for 24 h). However, pD2 values were not modified (10.78 +/- 0.03 and 5.62 +/- 0.04 for BK and carbachol, respectively) suggesting that no change in the apparent receptor affinity occurred. Thus, TNF alpha induced-alterations in Ca2+ homeostasis in human TSMC may be a key mechanism underlying airway hyperreactivity.

MeSH terms

  • Bradykinin / pharmacology*
  • Bradykinin / physiology
  • Calcium / metabolism*
  • Carbachol / pharmacology*
  • Cells, Cultured
  • Humans
  • Muscle, Smooth / drug effects*
  • Muscle, Smooth / physiology
  • Second Messenger Systems / drug effects
  • Second Messenger Systems / physiology
  • Trachea / drug effects*
  • Trachea / physiology
  • Tumor Necrosis Factor-alpha / pharmacology*
  • Tumor Necrosis Factor-alpha / physiology

Substances

  • Tumor Necrosis Factor-alpha
  • Carbachol
  • Bradykinin
  • Calcium