Targeted mutagenesis identifies Asp-569 as a catalytically critical residue in T7 RNA polymerase

Mol Gen Genet. 1995 Apr 10;247(1):110-3. doi: 10.1007/BF00425827.

Abstract

In order to look more closely at a well-conserved region in T7 RNA polymerase (T7 RNAP) containing, as shown earlier, the functionally essential residues Pro-563 and Tyr-571, we used targeted mutagenesis to change those residues within this region that are invariant in all single-subunit RNA polymerases, and characterized the mutant enzymes in vitro. The most interesting finding of this study was the crucial importance of the acidic group of Asp-569. In addition, we have shown that the phenolic ring is the most significant functional group of Tyr-571, with the hydroxy group also contributing to promoter binding.

MeSH terms

  • Amino Acid Sequence
  • Aspartic Acid / physiology*
  • Bacteriophage T7 / enzymology*
  • DNA-Binding Proteins / chemistry
  • DNA-Directed RNA Polymerases / chemistry*
  • DNA-Directed RNA Polymerases / metabolism
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Promoter Regions, Genetic
  • Structure-Activity Relationship
  • Transcription, Genetic
  • Tyrosine / physiology
  • Viral Proteins

Substances

  • DNA-Binding Proteins
  • Viral Proteins
  • Aspartic Acid
  • Tyrosine
  • bacteriophage T7 RNA polymerase
  • DNA-Directed RNA Polymerases